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(1) “Enantioselective Synthesis of Bicyclo[2.2.2]octenones Using a Copper-Mediated Oxidated Dearomatization/[4+2] Dimerization Cascade," Dong, S.; Zhu, J.; Porco, J. A., Jr.J. Am. Chem. Soc., 2008, 130, 2738-2739.
[ Link to Publication ]
(2) “Preparation of Alkylidene Indane and Related Scaffolds and Their Further Elaboration to Novel Chemotypes," Kesavan, S.; Panek, J. S.; Porco, J. A., Jr.Org. Lett., 2007, 9, 5203-5206.
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(3) “1,2-Dihydroisoquinolines as Templates for Cascade Reactions to Access Isoquinoline Alkaloid Frameworks," Su, S.; Porco, J. A., Jr.Org. Lett., 2007, 9, 4983-4986.
[ Link to Publication ]
(4) “Identification of Novel Epoxide Inhibitors of Hepatitis C Virus Replication Using a High-Throughput Screen," Peng, L. F.; Kim, S. S.; Matchacheep, S.; Lei, X.; Su, S.; Lin, W.; Runguphan, W.; Choe, W. H.; Sakamoto, N.; Ikeda, M.; Kato, N.; Beeler, A. B.; Porco, J. A., Jr.; Schreiber, S. L.; Chung, R. T.Anti. Agents and Chemo., 2007, 51, 3756-3759.
[ Link to Publication ]
(5) “Nucleophilic Addition to N-Phosphinylimines Via Rare Earth Metal Triflate/Trifluoroacetic Anhydride Activation," Ong, W.W.; Beeler, A.B.; Kesavan, S.; Panek, J. S.; Porco, J. A., Jr.Angewandte Chemie International Edition, 2007, 46, 7470-7472.
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(6) “Skeletal Diversity through Radical Cyclization of Tetrahydropyridine Scaffolds," Dandapani, S.; Duduta, M.; Panek, J. S.; Porco, J. A., Jr.Org. Lett., 2007, 9, 3849-3852.
[ Link to Publication ]
(7) “Synthesis of Pyrrolo-isoquinolines Related to the Lamellarins Using Silver-Catalyzed Cycloisomerizaton/Dipolar Cycloaddition," Su, S.; Porco, J. A., Jr.J. Am. Chem. Soc., 2007, 129, 7744-7745.
[ Link to Publication ]
(8) “1,2,3,4-Tetrahydro-1,5-naphthyridines and related heterocyclic scaffolds: Exploration of suitable chemistry for library development," Woo, G.H.C.; Beeler, A.B.; Snyder, J.K.Tetrahedron, 2007, 63, 5649-5655.
[ Link to Publication ]
(9) “An Approach to Skeletal Diversity Using Functional Group Pairing of Multifunctional Scaffolds," Comer, E.; Rohan, E.; Deng, L.; Porco, J. A., Jr.Org. Lett., 2007, 9, 2123-2126.
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(10) “Stereochemical and Skeletal Diversity Employing Pipecolate Ester Scaffolds," Chen, Y.; Porco, J. A., Jr.; Panek, J. S.Org. Lett., 2007, 9, 1529-1532.
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(11) “Synthesis of Carbamates and Ureas Using Zr(IV)-Catalyzed Exchange Processes," Han, C.; Porco, J. A., Jr.Org. Lett., 2007, 9, 1517-1520.
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(12) “Synthesis of 5,6,7,8-Tetrahydro-1,6-naphthyridines and Related Heterocycles by Cobalt-Catalyzed [2 + 2 + 2] Cyclizations," Zhou, Y.; Porco, J. A., Jr.; Snyder, J. K. Org. Lett., 2007, 9, 393-396.
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(13) “Discovery of Chemical Reactions through Multidimensional Screening," Beeler, A. B.; Su, S.; Singleton, C. A.; Porco, J. A., Jr. J. Am. Chem. Soc., 2007, 129, 1413-1419.
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(14) “Convergent Synthesis of Complex Diketopiperazines Derived from Pipecolic Acid Scaffolds and Parallel Screening against GPCR Targets," Dandapani, S.; Lan, P.; Beeler, A. B.; Beischel, S.; Abbas, A.; Roth, B. L., Porco, J. A.,Jr.; Panek, J. S. J. Org. Chem., 2006, 71, 8934-8945.
[ Link to Publication ]
(15) “Asymmetric Allylboration of Ketones Catalyzed by Chiral Diols," Lou, S.; Moquist, P. N.; Schaus, S. E. J. Am. Chem. Soc., 2006, 128, 12660-12661.
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(16) “Exploring Skeletal Diversity via Ring Contraction of Glycal-Derived Scaffolds," Yeager, A. R.; Min, G. K.; Porco, J. A., Jr.; Schaus, S. E. Org. Lett., 2006, 8(22), 5065-5068.
[ Link to Publication ]
(17) “Enantioselective Synthesis of Linear Polypropionate Arrays Using Anthracene-Tagged Organosilanes ," Kesavan, S.; Su, Q.; Shao, J.; Porco, J. A., Jr.; Panek, J. S. Org. Lett., 2005, 7, 4435-4438.
[ Link to Publication ]
(18) “A new, chiral anthracene for the Diels-Alder/retro-Diels-Alder sequence in lactam and butenolide synthesis ," Sanyal, A.; Yuan, Q.; Snyder, J. K.Tetrahedron Lett., 2005, 46, 2475-2478.
[ Link to Publication ]
(19) “Chiral Anthracene and Anthrone templates as Stereocontrolling Elements in Diels-Alder/Retro Diels-Alder Sequences ," Burgess, K. l.; Corbett, M. S.; Eugenio, P.; Lajkiewicz; N. J.; Liu, X.; Sanyal, A.; Yan, W.; Yuan, Q.; Snyder, J. K.Bioorg, Med. Chem., 2005, 13, 5299-5309.
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(20) “Asymmetric Mannich Reactions of ß- Keto Esters with Acyl Imines Catalyzed by Cinchona Alkaloids ," Lou, Shao; Taoka, M. Brandon; Ting, Amal; Schaus, S. E. J. Am. Chem. Soc. , 2005, 127, 11256-11257.
[ Link to Publication ]
(21) “Chemical Library Synthesis Using Convergent Approaches," Beeler, A. B.; Schaus, S. E.; Porco, J. A., Jr. Curr. Opin. Chem. Bio., 2005, 9, 277-284.
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(22) “Synthesis of a Library of Complex Macrodiolides Employing Cyclodimerization of Hydroxy Esters," Beeler, A. B.; Acquilano, D. E.; Su, Q.; Yan, F.; Roth, B. L.; Panek, J. S.; Porco, J. A., Jr. J. Comb. Chem., 2005, 7, 673-681.
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(23) “Stereocontrolled Synthesis of a Complex Library via Elaboration of Angular Epoxyquinol Scaffolds," Lei, X.; Zaarur, N.; Sherman, M. Y.; Porco, J. A., Jr. J. Org. Chem., 2005, 70, 6474-6483.
[ Link to Publication ]
(24) “Convergent Synthesis of a Complex Oxime Library Using Chemical Domain Shuffling," Su, S.; Acquilano, D. E.; Arumugasamy, J.; Beeler, A. B.; Eastwood, E. L.; Giguere, J. R.; Lan, P.; Lei, X.; Min, G. K.; Yeager, A. R.; Zhou, Y.; Panek, J. S.; Snyder, J. K.; Schaus, S. E.; Porco, J. A., Jr. Org. Lett., 2005, 7, 2751-2754.
[ Link to Publication ]
(25) “Synthesis of a Polymer-Supported Anthracene and Its Application as a Dienophile Scavenger,” Lei, X.; Porco, J. A., Jr.; Org. Lett. 2004, 6, 795-798.
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(26) “Intramolecular Inverse-Electron-Demand Diels-Alder Reactions of Imidazoles with 1,2,4-Triazines : A New Route to 1,2,3,4-Tetrahydro-1,5-naphthyridines and Related Heterocycles,” Lahue, R. B.; Lo, Sie-Mun; Woo, H. C. Grace; Snyder, J. K. J. Org. Chem., 2004, 69, 7171- 7182.
[ Link to Publication ]
(27) “Synthesis of Complex Alkoxyamines Using a Polymer-Supported N-Hydroxyphthalimide,” Su, S.; Giguere, J. R.; Schaus, S. E.; Porco, J. A., Jr. Tetrahedron. 2004, 60, 8645-8657.
[ Link to Publication ]
(28) “Stereochemical Diversity through Cyclodimerization : Synthesis of Polyketide-like Macrodiolides,” Su, Q.; Beeler, A. B.; Lobkovsky, E.; Porco, J.A., Jr.; Panek, J. S. Organic Lett. 2003, 5, 2149-2152.
[ Link to Publication ]
(29) "The Development of a Chromatography-Free Mitsunobu Reaction : Synthesis and Applications of an Anthracene-Tagged Phosphine Reagent,” Lan, P.; Porco, J. A., Jr.; South, M. S.; Parlow, J. J. J. Comb. Chem. 2003, 5, 660-669.
[ Link to Publication ]
(30) “Polymer-Assisted Solution-Phase (PASP) Suzuki Couplings Employing an Anthracene-Tagged Palladium Catalyst,” Lan, P.; Berta, D.; Porco, J. A., Jr.; South, M. S.; Parlow, J. J. J. Org. Chem. 2003, 68, 9678-9686.
[ Link to Publication ]
(31) “Combinatorial Synthesis of Natural Product-like Molecules Using a First Generation Spiroketal Scaffold,” Kulkarni, B.A.; Roth, G. P.; Lobkovsky, E.; Porco, J. A., Jr. J. Comb. Chem. 2002, 4, 56-72.
[ Link to Publication ]
(32) “Parallel Synthesis and Purification using Anthracene-Tagged Substrates,” Wang, X.; Parlow, J. J.; Porco, J.A., Jr. Organic Lett. 2000, 2, 3509-3512.
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